PSN632408 | GPR119 agonist | Probechem Biochemicals

Chemical Structure : PSN632408

CAS No.: 857652-30-3

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PSN632408 (PSN 632408)

货号: PC-20444Not For Human Use, Lab Use Only.

PSN632408 (PSN 632408) is a selective small-molecule GPR119 agonist with cAMP EC50 of 7.9 and 5.6 uM for mouse and human GPR119 receptor, respectively.

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5 mg	￥780	In stock
10 mg	￥1180	In stock
25 mg	￥2180	In stock
50 mg	￥3680	In stock
100 mg		Get quote

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生物&药学活性

PSN632408 (PSN 632408) is a selective small-molecule GPR119 agonist with cAMP EC50 of 7.9 and 5.6 uM for mouse and human GPR119 receptor, respectively.
PSN632408 is selective for GPR119, shows no acitvities against cannabinoid receptors CB1 and CB2, PPARα, PPARγ, as well as a set of 107 targets comprising GPCRs, ligand-gated ion channels, other receptors.
PSN632408 (30-100 mg/kg, i.p.) acutely reduce food intake in freely feeding male Sprague-Dawley rats, did not significantly alter locomotor activity.
PSN632408 (100 mg, Oral) reduces body weight gain and white adipose tissue deposition upon subchronic oral administration to high-fat-fed rats.

物理化学性质&存储条件

分子量	360.41
分子式	C18H24N4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	tert-butyl 4-((3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl)methoxy)piperidine-1-carboxylate

参考文献

1. Overton HA,, et al. Cell Metab. 2006 Mar;3(3):167-75.

PSN632408 (PSN 632408)

生物&药学活性

物理化学性质&存储条件

参考文献

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PSN632408 (PSN 632408)

生物&药学活性

物理化学性质&存储条件

参考文献

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