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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Pyruvate Dehydrogenase Kinase (PDK)-PS10
PS10

Chemical Structure : PS10

CAS No.: 1564265-82-2

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PS10 (PDK inhibitor PS10)

货号: PC-63500Not For Human Use, Lab Use Only.

PS10 (PDK inhibitor PS10) is a novel potent and highly selective pyruvate dehydrogenase kinase (PDK) inhibitor with IC50 values of 0.8 μM, 0.76 μM, 2.1 μM and 21.3 μM for PDK2, PDK4, PDK1, and PDK3, respectively.

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5 mg ￥780 In stock
10 mg ￥1180 In stock
25 mg ￥1980 In stock
50 mg ￥3280 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

PS10 (PDK inhibitor PS10) is a novel potent and highly selective pyruvate dehydrogenase kinase (PDK) inhibitor with IC50 values of 0.8 μM, 0.76 μM, 2.1 μM and 21.3 μM for PDK2, PDK4, PDK1, and PDK3, respectively.
PS10 improved glucose tolerance, stimulates myocardial carbohydrate oxidation in diet-induced obesity.
PS10 is a more suitable PDK inhibitor for treatment of diabetic cardiomyopathy.

物理化学性质&存储条件

分子量 323.319
分子式 C14H13NO6S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-[(2,4-dihydroxyphenyl)sulfonyl] isoindoline-4,6-diol

参考文献

1. Wu CY, et al. J Biol Chem. 2018 May 8. pii: jbc.RA118.002838.

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