PK-THPP

Chemical Structure : PK-THPP

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货号: PC-20698Not For Human Use, Lab Use Only.

TASK-3 inhibitor 23 is a potent, selective inhibitor of TWIK-related acid-sensitive K+ (K2P9.1, TASK-3) ion channel with IC50 of 30 nM, 10-fold selectivity over TASK-1.

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生物&药学活性

PK-THPP is a potent, selective inhibitor of TWIK-related acid-sensitive K+ (K2P9.1, TASK-3) ion channel with IC50 of 30 nM, 10-fold selectivity over TASK-1.
PK-THPP demonstrated pharmacological target engagement as indicated by its ability to modulate sleep architecture in rodent electroencephalogram (EEG) telemetry models.

物理化学性质&存储条件

分子量	468.60
分子式	C29H32N4O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	CCCC(C1CCN(C2=C(CN(C(C3=CC=C(C4=CC=CC=C4)C=C3)=O)CC5)C5=NC=N2)CC1)=O

参考文献

1. Craig A Coburn, et al. ChemMedChem. 2012 Jan 2;7(1):123-33.

PK-THPP

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PK-THPP

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