PFI-5 | SMYD2 inhibitor | Probechem Biochemicals

Chemical Structure : PFI-5

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PFI-5 (SMYD2 inhibitor PFI-5, PFI5)

货号: PC-73054Not For Human Use, Lab Use Only.

PFI-5 a highly biochemically potent, selective, and cell-active SMYD2 chemical probe with IC50 of 8 nM.

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100 mg		Get quote

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生物&药学活性

PFI-5 a highly biochemically potent, selective, and cell-active SMYD2 chemical probe with IC50 of 8 nM.
PFI-5 inhibits p53 methylation in MCF7 cells with EC50 of 1.3 uM, with no toxicity.

物理化学性质&存储条件

分子量	501.679
分子式	C29H39N7O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-(3-(4-amino-6-methyl-1H-imidazo[4,5-c]pyridin-1-yl)-3-methylazetidin-1-yl)(1-((1-(cyclohept-2-en-1-yl)piperidin-4-yl)methyl)-1H-pyrrol-3-yl)methanone

参考文献

1. Taylor AP, et al. J Med Chem. 2019 Sep 12;62(17):7669-7683.

PFI-5 (SMYD2 inhibitor PFI-5, PFI5)

生物&药学活性

物理化学性质&存储条件

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PFI-5 (SMYD2 inhibitor PFI-5, PFI5)

生物&药学活性

物理化学性质&存储条件

参考文献

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