PF-CBP1 hydrochloride |CAS: 2070014-93-4 Probechem Biochemicals

Chemical Structure : PF-CBP1 hydrochloride

CAS No.: 2070014-93-4

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PF-CBP1 hydrochloride (PF CBP1 hydrochloride)

货号: PC-45780Not For Human Use, Lab Use Only.

PF-CBP1 hydrochloride is a potent, highly selective inhibitor of the CBP and p300 bromodomains with IC50 of 125 nM and 363 nM, respectively.

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10 mg	￥880	In stock
25 mg	￥1380	In stock
50 mg	￥2180	In stock
100 mg	￥3680	In stock
200 mg		Get quote
1 g		Get quote

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生物&药学活性

PF-CBP1 hydrochloride is a potent, highly selective inhibitor of the CBP and p300 bromodomains with IC50 of 125 nM and 363 nM, respectively.
PF-CBP1 displays >100-fold selectivity for the bromodomain of CBP over those of BRD4 and a panel of other proteins.
PF-CBP1 reduces the expression of inflammatory cytokines by LPS-stimulated primary macrophages, also suppresses the expression of RGS4 in primary cortical neurons.

物理化学性质&存储条件

分子量	525.0821
分子式	C29H37ClN4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	DMSO: ≥ 34 mg/mL
Chemical Name/SMILES	4-(2-(5-(3,5-dimethylisoxazol-4-yl)-2-(4-propoxyphenethyl)-1H-benzo[d]imidazol-1-yl)ethyl)morpholine hydrochloride

参考文献

1. Chekler EL, et al. Chem Biol. 2015 Dec 17;22(12):1588-96.

PF-CBP1 hydrochloride (PF CBP1 hydrochloride)

生物&药学活性

物理化学性质&存储条件

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PF-CBP1 hydrochloride (PF CBP1 hydrochloride)

生物&药学活性

物理化学性质&存储条件

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