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首页-小分子抑制剂&激动剂-GPCR-Cannabinoid Receptor-PF-514273
PF-514273

Chemical Structure : PF-514273

CAS No.: 851728-60-4

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PF-514273 (PF 514273)

货号: PC-20521Not For Human Use, Lab Use Only.

PF-514273 (PF 514273) is a potent, selective and orally active antagonist of cannabinoid CB1 receptor with Ki of 1.0 nM, >10000-fold selectivity for CB1 over CB2.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

PF-514273 (PF 514273) is a potent, selective and orally active antagonist of cannabinoid CB1 receptor with Ki of 1.0 nM, >10000-fold selectivity for CB1 over CB2.

物理化学性质&存储条件

分子量 452.28
分子式 C21H17Cl2F2N3O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

O=C1N(CC(F)(F)C)CCOC2=C(C3=CC=C(Cl)C=C3)N(C4=CC=CC=C4Cl)N=C12

参考文献

1. Dow RL, et al. J Med Chem. 2009 May 14;52(9):2652-5.

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