PF-4363467 |CAS:2040055-84-1 Probechem Biochemicals

Chemical Structure : PF-4363467

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PF-4363467 (PF 04363467;PF4363467)

货号: PC-61108Not For Human Use, Lab Use Only.

PF-4363467 (PF 04363467) is a novel highly potent, brain penetrant dopamine D3/D2 receptor antagonist with Ki of 1.3/692 nM respectively, with high selectivity for D3R versus other biogenic amine receptors.

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生物&药学活性

PF-4363467 (PF 04363467) is a novel highly potent, brain penetrant dopamine D3/D2 receptor antagonist with Ki of 1.3/692 nM respectively, with high selectivity for D3R versus other biogenic amine receptors; dose-dependently attenuated opioid self-administration and opioid drug-seeking behavior in a rat operant reinstatement model using animals trained to self-administer fentanyl.

物理化学性质&存储条件

分子量	402.553
分子式	C22H30N2O3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-N-(4-(4-ethylmorpholin-2-yl)-2-methylphenyl)-4-isopropylbenzenesulfonamide

参考文献

1. Wager TT, et al. ACS Chem Neurosci. 2017 Jan 18;8(1):165-177.

PF-4363467 (PF 04363467;PF4363467)

生物&药学活性

物理化学性质&存储条件

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PF-4363467 (PF 04363467;PF4363467)

生物&药学活性

物理化学性质&存储条件

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