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首页-小分子抑制剂&激动剂-GPCR-Glucagon Receptor-PF-07976016
PF-07976016

Chemical Structure : PF-07976016

CAS No.: 3059496-70-4

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PF-07976016 (PF07976016)

货号: PC-28066Not For Human Use, Lab Use Only.

PF-07976016 is a potent, orally active glucose-dependent insulinotropic polypeptide receptor (GIPR) antagonist with IC50 of 4.1 nM, shows competitively binding to GIPR and blocking the increase in Gαs-mediated cAMP production induced by GIP agonists.

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10 mg ￥780 In stock
25 mg ￥1280 In stock
50 mg ￥1980 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

PF-07976016 is a potent, orally active glucose-dependent insulinotropic polypeptide receptor (GIPR) antagonist with IC50 of 4.1 nM, shows competitively binding to GIPR and blocking the increase in Gαs-mediated cAMP production induced by GIP agonists.

物理化学性质&存储条件

分子量 471.56
分子式 C28H29N3O4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(R)-4'-(1-((4-Isopropylphenyl)carbamoyl)pyrrolidine-2-carboxamido)-[1,1'-biphenyl]-4-carboxylic acid

参考文献

1. Patent WO2024214038 A1 2024-10-17.

2. Patent US20250235460 A1.

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