PF-03550096 | CB2 agonist | Probechem Biochemicals

Chemical Structure : PF-03550096

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PF-03550096 (PF03550096)

货号: PC-26032Not For Human Use, Lab Use Only.

PF-03550096 is a potent, selective orally active cannabinoid receptor 2 (CB2) agonist with Ki of 7.9 nM and 47 nM for human and rat CB2 receptors respectively.

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生物&药学活性

PF-03550096 is a potent, selective orally active cannabinoid receptor 2 (CB2) agonist with Ki of 7.9 nM and 47 nM for human and rat CB2 receptors respectively.
PF-03550096 is a full agonist and showed high selectivity for human CB(2) receptors in cell-based functional assay.
Orally administered PF-03550096 (3, 10 mg/kg) inhibited the 2,4,6-trinitrobenzene sulfonic acid (TNBS)-induced decrease in colonic pain threshold with statistical significance.

物理化学性质&存储条件

分子量	376.46
分子式	C19H28N4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-[(1S)-1-(aminocarbonyl)-2,2-dimethylpropyl]-3-(3-hydroxy-3-methylbutyl)-2-oxo-2,3-dihydro-1H-benzimidazole-1-carboxamide

参考文献

1. Akira Kikuchi, et al. J Pharmacol Sci. 2008 Feb;106(2):219-24.

PF-03550096 (PF03550096)

生物&药学活性

物理化学性质&存储条件

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PF-03550096 (PF03550096)

生物&药学活性

物理化学性质&存储条件

参考文献

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