PELI1-IN-1 | PELI1 inhibitor | Probechem Biochemicals

Chemical Structure : PELI1-IN-1

CAS No.: 3034889-94-3

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PELI1-IN-1 (Compound 3d)

货号: PC-26725Not For Human Use, Lab Use Only.

PELI1-IN-1 (PELI1 inhibitor 3d) is a specific small molecule inhibitor of E3 ubiquitin ligase Pellino-1 (PELI1) with binding Kd of 8.2 uM in fluorescence quenching assays, interrupts the interaction of PELI1 and SNAIL/SLUG.

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10 mg	￥5280	In stock
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生物&药学活性

PELI1-IN-1 (PELI1 inhibitor 3d) is a specific small molecule inhibitor of E3 ubiquitin ligase Pellino-1 (PELI1) with binding Kd of 8.2 uM in fluorescence quenching assays, interrupts the interaction of PELI1 and SNAIL/SLUG.
PELI1-IN-1 exhibits potent anti-TNBC activity against cell migration without affecting cell proliferation in vitro.
PELI1-IN-1 shows potent anti-TNBC metastasis efficacy without observable toxic side effects in vivo.

物理化学性质&存储条件

分子量	320.34
分子式	C20H16O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-3'-(3,5-dihydroxystyryl)-[1,1'-biphenyl]-3,4'-diol

参考文献

1. Guangsen Xu, et al. Eur J Med Chem. 2023 Dec 20:265:116060.

PELI1-IN-1 (Compound 3d)

生物&药学活性

物理化学性质&存储条件

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PELI1-IN-1 (Compound 3d)

生物&药学活性

物理化学性质&存储条件

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