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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Calpain-PD150606
PD150606

Chemical Structure : PD150606

CAS No.: 179528-45-1

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PD150606 (PD 150606, PD-150606)

货号: PC-42190Not For Human Use, Lab Use Only.

PD150606 is a potent and selective calpain inhibitor with Ki of 0.21 uM/0.37 uM for u-calpain/m-calpain, respectively.

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10 mg ￥980 In stock
25 mg ￥1580 In stock
50 mg ￥2680 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

PD150606 is a potent and selective calpain inhibitor with Ki of 0.21 uM/0.37 uM for u-calpain/m-calpain, respectively.
PD150606 shows no inhibition for other proteases (cathepin B, papain, trypsin and thermolysin (Ki> 500 uM).
PD150606 attenuate shypoxic/hypoglycemic injury to cerebrocortical neurons in culture and excitotoxic injury to Purkinje cells in cerebellar slices.

物理化学性质&存储条件

分子量 306.1201
分子式 C9H7IO2S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: ≥ 28 mg/mL
Chemical Name/SMILES

2-Propenoic acid, 3-(4-iodophenyl)-2-mercapto-, (2Z)-

参考文献

1. Wang KK, et al. Proc Natl Acad Sci U S A. 1996 Jun 25;93(13):6687-92.

2. Niapour M, et al. J Biol Chem. 2008 Aug 1;283(31):21371-81.

3. Waters SL, et al. J Pharmacol Exp Ther. 1997 Dec;283(3):1177-84.

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