PCSK9 inhibitor 9 |CAS:2215931-60-3 Probechem Biochemicals

Chemical Structure : PCSK9 inhibitor 9

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PCSK9 inhibitor 9

货号: PC-38279Not For Human Use, Lab Use Only.

PCSK9 inhibitor 9 is a small-molecule ligand with high affinity for a novel allosteric binding site on PCSK9.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

PCSK9 inhibitor 9 is a small-molecule ligand with high affinity for a novel allosteric binding site on PCSK9.
PCSK9 inhibitor 9 showed good target engagement with PCSK9 in Huh7 cell lysate.

物理化学性质&存储条件

分子量	631.719
分子式	C34H34FN3O6S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2'-fluoro-4'-(((1R)-1-methyl-1-(2-oxo-2-(thiazol-2-ylamino)ethyl)-6-((tetrahydro-2H-pyran-2-yl)methoxy)-1,2,3,4-tetrahydroisoquinolin-7-yl)oxy)-[1,1'-biphenyl]-4-carboxylic acid

参考文献

1. Whitney L Petrilli, et al. Cell Chem Biol. 2020 Jan 16;27(1):32-40.e3.