Otamixaban |CAS:193153-04-7 Probechem Biochemicals

Chemical Structure : Otamixaban

CAS No.: 193153-04-7

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Otamixaban (FXV-673)

货号: PC-45940Not For Human Use, Lab Use Only.

A potent and selective factor Xa (FXa) inhibitor with Ki of 0.4 nM.

规格	价格	库存	数量
100 mg	￥9872.0	In stock

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生物&药学活性

A potent and selective factor Xa (FXa) inhibitor with Ki of 0.4 nM; shows >1,000-fold selectivity over thrombin, activated protein C (aPC), plasmin, and tissue-plasminogen activator (t-PA); dose-dependently prolongs the time to vessel occlusion and inhibits thrombus formation in canine models of thrombosis.

Thrombosis

Phase 3 Discontinued

物理化学性质&存储条件

分子量	446.4984
分子式	C25H26N4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzenepropanoic acid, 3-(aminoiminomethyl)-.alpha.-[(1R)-1-[[4-(1-oxido-4-pyridinyl)benzoyl]amino]ethyl]-, methyl ester, (.alpha.R)-

参考文献

1. Guertin KR, et al. Bioorg Med Chem Lett. 2002 Jun 17;12(12):1671-4.

2. Chu V, et al. Thromb Res. 2001 Aug 15;103(4):309-24.

3. Rebello SS, et al. J Cardiovasc Pharmacol. 2001 Aug;38(2):288-97.

Otamixaban (FXV-673)

生物&药学活性

物理化学性质&存储条件

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Otamixaban (FXV-673)

生物&药学活性

物理化学性质&存储条件

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