Org 27569 |CAS:868273-06-7 Probechem Biochemicals

Chemical Structure : Org 27569

CAS No.: 868273-06-7

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Org 27569 (Org-27569;Org27569)

货号: PC-43465Not For Human Use, Lab Use Only.

Org 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor, significantly increases the binding of the CB1 receptor agonist [3H]CP 55,940 with pKb of 5.67.

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10 mg	￥780	In stock
25 mg	￥1380	In stock
50 mg	￥2280	In stock
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生物&药学活性

Org 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor, significantly increases the binding of the CB1 receptor agonist [3H]CP 55,940 with pKb of 5.67.
Org 27569 reduces food consumption in rats, produces CB1-independent hypophagic effects and does not affect the discriminative stimulus effects of anandamide (AEA).

物理化学性质&存储条件

分子量	409.95
分子式	C24H28ClN3O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 52.2 mg/mL
Chemical Name/SMILES	1H-Indole-2-carboxamide, 5-chloro-3-ethyl-N-[2-[4-(1-piperidinyl)phenyl]ethyl]-

参考文献

1. Price MR, et al. Mol Pharmacol. 2005 Nov;68(5):1484-95.

2. Erdozain AM, et al. Biochem Pharmacol. 2012 Jan 15;83(2):260-8.

3. Fay JF, et al. J Biol Chem. 2012 Sep 28;287(40):33873-82.

4. Gamage TF, et al. Behav Pharmacol. 2014 Apr;25(2):182-5.

Org 27569 (Org-27569;Org27569)

生物&药学活性

物理化学性质&存储条件

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Org 27569 (Org-27569;Org27569)

生物&药学活性

物理化学性质&存储条件

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