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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Dipeptidyl Peptidase (DPP)-Omarigliptin
Omarigliptin

Chemical Structure : Omarigliptin

CAS No.: 1226781-44-7

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Omarigliptin (MK-3102, MK3102)

货号: PC-44866Not For Human Use, Lab Use Only.

Omarigliptin (MK-3102) is a potent and selective DPP-4 inhibitor with IC50 of 1.4 nM.

规格 价格 库存 数量
10 mg ￥1280 In stock
25 mg ￥1980 In stock
50 mg ￥2980 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Omarigliptin (MK-3102) is a potent and selective DPP-4 inhibitor with IC50 of 1.4 nM.
Omarigliptin (MK-3102) shows high selectivity against QPP, DPP8,FAP (IC50>20 uM).
Omarigliptin (MK-3102) is efficacious in the diabetes PD model and excellent pharmacokinetic profile.

物理化学性质&存储条件

分子量 398.4275
分子式 C17H20F2N4O3S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2H-Pyran-3-amine, 2-(2,5-difluorophenyl)-5-[2,6-dihydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-, (2R,3S,5R)-

参考文献

1. Biftu T, et al. Bioorg Med Chem Lett. 2013 Oct 1;23(19):5361-6.

2. Biftu T, et al. J Med Chem. 2014 Apr 24;57(8):3205-12.

3. Burness CB. Drugs. 2015 Nov;75(16):1947-52.

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