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首页-小分子抑制剂&激动剂-GPCR-Cannabinoid Receptor-Olorinab
Olorinab

Chemical Structure : Olorinab

CAS No.: 1268881-20-4

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Olorinab (APD371, APD-371)

货号: PC-60146Not For Human Use, Lab Use Only.

Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM.

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5 mg ￥1280 In stock
10 mg ￥1980 In stock
25 mg ￥3580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM.
Olorinab (APD371) displays no activity against CB1 receptors (EC50>10 uM).
Olorinab (APD371) exhibits activity in rat model of osteoarthritis pain.

物理化学性质&存储条件

分子量 357.414
分子式 C18H23N5O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

3-((4aS,5aS)-3-(((S)-1-hydroxy-3,3-dimethylbutan-2-yl)carbamoyl)-4,4a,5,5a-tetrahydro-1H-cyclopropa[4,5]cyclopenta[1,2-c]pyrazol-1-yl)pyrazine 1-oxide

参考文献

1. Sangdon Han, et al. ACS Med. Chem. Lett., 2017, 8 (12), pp 1309-1313.

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