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首页-小分子抑制剂&激动剂-GPCR-Dopamine Receptor-OS-3-106
OS-3-106

Chemical Structure : OS-3-106

CAS No.: 1580000-17-4

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OS-3-106 (Dopamine D3 receptor agonist)

货号: PC-38469Not For Human Use, Lab Use Only.

OS-3-106 is a high-affinity, selective dopamine D3 receptor (D3R) partial agonist with Ki value of 0.2 nM, exhibits 115-fold binding selectivity for D3R compared with the D2R.

规格 价格 库存 数量
10 mg ￥980 In stock
25 mg ￥1580 In stock
50 mg ￥2680 In stock
100 mg ￥4580 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

OS-3-106 is a high-affinity, selective dopamine D3 receptor (D3R) partial agonist with Ki value of 0.2 nM, exhibits 115-fold binding selectivity for D3R compared with the D2R.
OS-3-106 is also a partial agonist at the D2R (47% of quinpirole).
OS-3-106 (10 mg/kg) reduced cocaine self-administration, also reduced responding for sucrose and locomotor activity.
OS-3-106 attenuated yawning induced by low doses of 7-OH-DPAT (a D3R-mediated behavior).

物理化学性质&存储条件

分子量 450.60
分子式 C25H30N4O2S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-[4-[4-(2-Methoxyphenyl)-1-piperazinyl]butyl]-4-(4-thiazolyl)benzamide

参考文献

1. Timothy H C Cheung, et al. J Pharmacol Exp Ther. 2013 Nov;347(2):410-23.

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