ORM-15341 (Ketodarolutamide, BAY1896953) | AR inhibitor

Chemical Structure : ORM-15341

CAS No.: 1297537-33-7

加入收藏

ORM-15341 (Ketodarolutamide, BAY1896953, ORM15341)

货号: PC-45612Not For Human Use, Lab Use Only.

ORM-15341 (Ketodarolutamide, BAY1896953) is the active main metabolite of ODM-201, a potent wt/mutant androgen receptor (AR) inhibitor, inhibits wtAR/AR(F876L) with IC50s of 25/51 nM respectively.

规格	价格	库存
10 mg	￥980	In stock
25 mg	￥1580	In stock
50 mg	￥2480	In stock
100 mg	￥3980	In stock
250 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

ORM-15341 (Ketodarolutamide, BAY1896953) is the active main metabolite of ODM-201, a potent wt/mutant androgen receptor (AR) inhibitor, inhibits wtAR/AR(F876L) with IC50s of 25/51 nM respectively.
ORM-15341 (Ketodarolutamide, BAY1896953) suppresses androgen-induced cell proliferation more efficaciously than enzalutamide or ARN-509.

物理化学性质&存储条件

分子量	396.8303
分子式	C19H17ClN6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 37 mg/mL
Chemical Name/SMILES	1H-Pyrazole-3-carboxamide, 5-acetyl-N-[(1S)-2-[3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl]-1-methylethyl]-

参考文献

1. Moilanen AM, et al. Sci Rep. 2015 Jul 3;5:12007.

ORM-15341 (Ketodarolutamide, BAY1896953, ORM15341)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

ORM-15341 (Ketodarolutamide, BAY1896953, ORM15341)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.