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首页-小分子抑制剂&激动剂-Epigenetics-Bromodomain-OF-1
OF-1

Chemical Structure : OF-1

CAS No.: 919973-83-4

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OF-1 (OF1, BRPF1 inhibitor)

货号: PC-62276Not For Human Use, Lab Use Only.

OF-1 is a potent bromodomain inhibitor that inhibits BRPF1B/2/3 bromodomains with Kd of 0.1/0.5/2.4 uM.

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5 mg ￥580 In stock
10 mg ￥880 In stock
25 mg ￥1380 In stock
50 mg ￥2180 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

OF-1 is a potent bromodomain inhibitor that inhibits BRPF1B/2/3 bromodomains with Kd of 0.1/0.5/2.4 uM; displays good selectivity against other bromodomains, 39-fold selectivity over closest off-target BRD4.

物理化学性质&存储条件

分子量 440.312
分子式 C17H18BrN3O4S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-bromo-N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methylbenzenesulfonamide

参考文献

1. Demont EH, et al. ACS Med Chem Lett. 2014 Sep 10;5(11):1190-5.

2. Pérez-Salvia M, et al. Epigenetics. 2017 May 4;12(5):323-339.

3. Meier JC, et al. ACS Chem Biol. 2017 Oct 20;12(10):2619-2630.

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