Nelotanserin (RVT-102, APD125) | 5-HT2A antagonist | Probechem Biochemicals

Chemical Structure : Nelotanserin

CAS No.: 839713-36-9

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Nelotanserin (APD-125, RVT-102, APD125, RVT102)

货号: PC-42651Not For Human Use, Lab Use Only.

Nelotanserin (RVT-102, APD125) is a potent, selective 5-HT2A inverse agonist with pKi of 9.2.

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5 mg	￥880	In stock
10 mg	￥1280	In stock
25 mg	￥2180	In stock
50 mg	￥3580	In stock
100 mg		Get quote

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生物&药学活性

Nelotanserin (RVT-102, APD125) is a potent, selective 5-HT2A inverse agonist with pKi of 9.2.
Nelotanserin displays >30- and 5000-fold selectivity compared with 5-HT2C and 5-HT2B receptors.
Nelotanserin prevents DOI-induced hypolocomotion and increases sleep consolidation; orally active.

物理化学性质&存储条件

分子量	437.2381
分子式	C18H15BrF2N4O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 32 mg/mL
Chemical Name/SMILES	Urea, N-[3-(4-bromo-1-methyl-1H-pyrazol-5-yl)-4-methoxyphenyl]-N'-(2,4-difluorophenyl)-

参考文献

1. Teegarden BR, et al. J Med Chem. 2010 Mar 11;53(5):1923-36.

2. Al-Shamma HA, et al. J Pharmacol Exp Ther. 2010 Jan;332(1):281-90.

Nelotanserin (APD-125, RVT-102, APD125, RVT102)

生物&药学活性

物理化学性质&存储条件

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Nelotanserin (APD-125, RVT-102, APD125, RVT102)

生物&药学活性

物理化学性质&存储条件

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