Nelfinavir mesylate |CAS:159989-65-8 Probechem Biochemicals

Chemical Structure : Nelfinavir mesylate

CAS No.: 159989-65-8

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Nelfinavir mesylate (AG-1343 mesylate, AG1343 mesylate)

货号: PC-44304Not For Human Use, Lab Use Only.

Nelfinavir (AG-1343) mesylate is a potent and orally bioavailable HIV-1 protease inhibitor with Ki of 2 nM.

规格	价格	库存
5 mg	￥980	In stock
10 mg	￥1580	In stock
50 mg	￥3280	In stock
100 mg		Get quote

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生物&药学活性

Nelfinavir (AG-1343) mesylate is a potent and orally bioavailable HIV-1 protease inhibitor with Ki of 2 nM.
Nelfinavir (AG-1343) exhibits an antiviral EC50 of 30 nM in HIV-1 strain RF-infected CEM-SS cells.
Nelfinavir (AG-1343) also inhibits the proliferation of NSCLC cells, as well as every cell line in the NCI60 cell line panel with mean GI50 of 5.2 uM, induces endoplasmic reticulum stress, autophagy, and apoptosis in vitro and in vivo.

物理化学性质&存储条件

分子量	663.8881
分子式	C33H49N3O7S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-, methanesulfonate (1:1)

参考文献

1. Zhang KE, et al. Antimicrob Agents Chemother. 2001 Apr;45(4):1086-93.

2. Shetty BV, et al. Antimicrob Agents Chemother. 1996 Jan;40(1):110-4.

3. Gills JJ, et al. Clin Cancer Res. 2007 Sep 1;13(17):5183-94.

Nelfinavir mesylate (AG-1343 mesylate, AG1343 mesylate)

生物&药学活性

物理化学性质&存储条件

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Nelfinavir mesylate (AG-1343 mesylate, AG1343 mesylate)

生物&药学活性

物理化学性质&存储条件

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