NTSR1 agonist RTI-3a

Chemical Structure : NTSR1 agonist RTI-3a

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货号: PC-28389Not For Human Use, Lab Use Only.

NTSR1 agonist RTI-3a is a potent, selective partial agonist of neurotensin receptor 1 (NTSR1) with EC50 of 67 nM and Emax of 54%.

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NTSR1 agonist RTI-3a is a potent, selective partial agonist of neurotensin receptor 1 (NTSR1) with EC50 of 67 nM and Emax of 54%.

分子量	522.99
分子式	C27H27ClN4O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(1-(7-chloroquinolin-4-yl)-5-(2,6-dimethoxyphenyl)-1H-pyrazole-3-carbonyl)-L-leucine

1. James B Thomas, et al. Bioorg Med Chem Lett. 2009 Mar 1;19(5):1438-41.