NTRC-824 | NTSR2 antagonist | Probechem Biochemicals

Chemical Structure : NTRC-824

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NTRC-824 (NTRC824)

货号: PC-22266Not For Human Use, Lab Use Only.

NTRC-824 is the first nonpeptide, selective antagonist of neurotensin receptor type 2 (NTS2/NTSR2) with IC50 of 32 nM in FLIPR assays, binding Ki of 202 nM.

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生物&药学活性

NTRC-824 is the first nonpeptide, selective antagonist of neurotensin receptor type 2 (NTS2/NTSR2) with IC50 of 32 nM in FLIPR assays, binding Ki of 202 nM.
NTRC-824 displays no significant affinity for NTS1 (Ki>30 uM).

物理化学性质&存储条件

分子量	553.55
分子式	C25H26F3N3O6S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-[(5-{[(4-methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-l-leucine

参考文献

1. Thomas JB, et al. J Med Chem. 2014 Sep 11;57(17):7472-7.

NTRC-824 (NTRC824)

生物&药学活性

物理化学性质&存储条件

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NTRC-824 (NTRC824)

生物&药学活性

物理化学性质&存储条件

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