NSD2 inhibitor PTD2 | NSD2 inhibitor | Probechem Biochemicals

Chemical Structure : NSD2 inhibitor PTD2

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NSD2 inhibitor PTD2 (Ac-Gly-Val-Nle-Arg-Ile-NH2)

货号: PC-28088Not For Human Use, Lab Use Only.

NSD2 inhibitor PTD2 is a peptide derived from histone H4 sequence and inhibitor for the histone methyltransferase WHSC1 (Nuclear receptor-binding SET domain protein 2, NSD2, MMSET) with SPR KD of 3.0 uM, IC50 of 22 uM and 3.2 uM for NSD2 and NSD3 respectively.

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NSD2 inhibitor PTD2 is a peptide derived from histone H4 sequence and inhibitor for the histone methyltransferase WHSC1 (Nuclear receptor-binding SET domain protein 2, NSD2, MMSET) with SPR KD of 3.0 uM, IC50 of 22 uM and 3.2 uM for NSD2 and NSD3 respectively.
PTD2 demonstrates no enzymatic inhibition against the entire panel of methyltransferases.

物理化学性质&存储条件

分子量	597.76
分子式	C27H51N9O6
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Sequence: Ac-Gly-Val-Nle-Arg-Ile-NH2

参考文献

1. Morrison MJ, et al. PLoS One. 2018 May 9;13(5):e0197082.

NSD2 inhibitor PTD2 (Ac-Gly-Val-Nle-Arg-Ile-NH2)

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物理化学性质&存储条件

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NSD2 inhibitor PTD2 (Ac-Gly-Val-Nle-Arg-Ile-NH2)

生物&药学活性

物理化学性质&存储条件

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