NS3861 |CAS: 216853-60-0 Probechem Biochemicals

Chemical Structure : NS3861

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NS3861 (NS-3861;NS 3861)

货号: PC-60819Not For Human Use, Lab Use Only.

A potent, subtype-selective α3β4 nAChR partial agonist with Ki of 0.62 nM.

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1 g		Get quote

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生物&药学活性

A potent, subtype-selective α3β4 nAChR partial agonist with Ki of 0.62 nM; selectively activates receptors containing β4- but not β2-subunits, shows no efficacy at α4β2 receptors and only marginal efficacy at α4β4 receptors expressed in oocytes; enhances fecal pellet expulsion in a dose-dependent manner in mice that received long-term, but not short-term, morphine treatment.

物理化学性质&存储条件

分子量	400.29
分子式	C12H14BrNS.C4H4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene fumarate

参考文献

1. Harpsøe K, et al. J Biol Chem. 2013 Jan 25;288(4):2559-70.

2. Gade AR, et al. J Pharmacol Exp Ther. 2016 Jun;357(3):520-8.

NS3861 (NS-3861;NS 3861)

生物&药学活性

物理化学性质&存储条件

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NS3861 (NS-3861;NS 3861)

生物&药学活性

物理化学性质&存储条件

参考文献

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