MU1656 |CAS 2768008-84-8 Probechem Biochemicals

首页-小分子抑制剂&激动剂-Epigenetics-Histone Methyltransferase (HMTase)-MU1656

Chemical Structure : MU1656

加入收藏

MU1656 (MU 1656)

货号: PC-38010Not For Human Use, Lab Use Only.

MU1656 (MU 1656 ) is a potent, highly selective inhibitor of histone methyltransferase DOT1L with IC50 of 2 nM.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

MU1656 (MU 1656 ) is a potent, highly selective inhibitor of histone methyltransferase DOT1L with IC50 of 2 nM.
MU1656 displays highly selectively against a panel of 37 methyltransferases.
MU1656 is more metabolically stable and significantly less toxic in vivo than pinometostat.

物理化学性质&存储条件

分子量	559.759
分子式	C32H45N7O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1R,2S,3S,5R)-3-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-5-((((1r,3S)-3-(2-(5-(tert-butyl)-1H-benzo[d]imidazol-2-yl)ethyl)cyclobutyl)(isopropyl)amino)methyl)cyclopentane-1,2-diol

参考文献

1. Khirsariya P, et al. J Med Chem. 2022 Apr 14;65(7):5701-5723.

联系我们 sales@probechem.com

MU1656 (MU 1656)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

MU1656 (MU 1656)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.