MRS8209

Chemical Structure : MRS8209

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货号: PC-23512Not For Human Use, Lab Use Only.

MRS8209 is a potent, peripheral subtype-selective 5-HT2B serotonin receptor antagonist with Ki of 4.27 nM (human 5-HT2B), shows reduced affinity at the m5-HT2BR and r5-HT2BR (100-fold and 10-fold).

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MRS8209 is a potent, peripheral subtype-selective 5-HT2B serotonin receptor antagonist with Ki of 4.27 nM (human 5-HT2B), shows reduced affinity at the m5-HT2BR and r5-HT2BR (100-fold and 10-fold).

物理化学性质&存储条件

分子量	466.28
分子式	C17H19IN6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(1R,2R,3S,4R,5S)-4-(6-(Cyclopentylamino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbonitrile

参考文献

1. Tosh DK, et al. J Med Chem. 2024 Nov 26. doi: 10.1021/acs.jmedchem.4c02174.

MRS8209

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MRS8209

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