MRS7232 | DAT inhibitor | Probechem Biochemicals

Chemical Structure : MRS7232

加入收藏

MRS7232 (MRS-7232)

货号: PC-22974Not For Human Use, Lab Use Only.

MRS7232 is an allosteric, non-competitive inhibitor of human dopamine transporter (DAT) with EC50 of 34 nM, and norepinephrine transporter (NET), also is a potent A3AR agonist with Ki of 14.5 nM.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

MRS7232 is an allosteric, non-competitive inhibitor of human dopamine transporter (DAT) with EC50 of 34 nM, and norepinephrine transporter (NET), also is a potent A3AR agonist with Ki of 14.5 nM.

物理化学性质&存储条件

分子量	473.93
分子式	C21H20ClN5O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Ethyl (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate

参考文献

1. Tosh DK, et al. J Med Chem. 2017 Apr 13;60(7):3109-3123.

MRS7232 (MRS-7232)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

MRS7232 (MRS-7232)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.