Chemical Structure : MRGPRX2 antagonist C9
CAS No.: 1274013-03-4
货号: PC-38068Not For Human Use, Lab Use Only.
MRGPRX2 antagonist C9 is a potent and selective MRGPRX2 inverse agonist (antagonist) with Ki of 43 nM.
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
5 mg | ¥880 | In stock | |
10 mg | ¥1280 | In stock | |
25 mg | ¥2180 | In stock | |
50 mg | Get quote | ||
100 mg | Get quote |
大包装,大折扣!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
MRGPRX2 antagonist C9 is a potent and selective MRGPRX2 inverse agonist (antagonist) with Ki of 43 nM.
MRGPRX2 antagonist C9 displays no antagonist activity towards NK1R or MRGPRX4.
MRGPRX2 antagonist C9 inhibits (R)-ZINC-3573-stimulated LAD2 human mast cell degranulation in a concentration-dependent manner.
分子量 | 275.344 | |
分子式 | C12H9N3OS2 | |
外观性状 | Solid | |
储存条件 |
|
|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
3-(thiazol-2-ylmethyl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one |
1. Can Cao, et al. Nature. 2021 Dec;600(7887):170-175.
备案号:沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright