MPC-3100 |CAS:958025-66-6 Probechem Biochemicals

Chemical Structure : MPC-3100

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MPC-3100 (MPC 3100;MPC3100)

货号: PC-60471Not For Human Use, Lab Use Only.

MPC-3100 is a novel potent, selective, orally bioavailable Hsp90 inhibitor with IC50 of 0.14 uM.

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生物&药学活性

MPC-3100 is a novel potent, selective, orally bioavailable Hsp90 inhibitor with IC50 of 0.14 uM.
MPC-3100 displays antiproliferative activity against a panel of cancer cell lines with IC50 of <1 uM.
MPC-3100 exhibits good in vitro profiles and a characteristic molecular biomarker signature of Hsp90 inhibition both in vitro and in vivo, shows significant antitumor effects in multiple human cancer xenograft models.

物理化学性质&存储条件

分子量	549.4
分子式	C22H25BrN6O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S)-1-[4-[2-[6-amino-8-[(6-bromo-1,3-benzodioxol-5-yl)thio]-9H-purin-9-yl]ethyl]-1-piperidinyl]-2-hydroxy-1-propanone

参考文献

1. Kim SH, et al. J Med Chem. 2012 Sep 13;55(17):7480-501.

2. Kim SH, et al. Bioorg Med Chem Lett. 2015 Nov 15;25(22):5254-7.

MPC-3100 (MPC 3100;MPC3100)

生物&药学活性

物理化学性质&存储条件

参考文献

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MPC-3100 (MPC 3100;MPC3100)

生物&药学活性

物理化学性质&存储条件

参考文献

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