MMSET-IN-1 |CAS:1998139-29-9 Probechem Biochemicals

首页-小分子抑制剂&激动剂-Epigenetics-Histone Methyltransferase (HMTase)-MMSET-IN-1

Chemical Structure : MMSET-IN-1

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MMSET-IN-1 (NSD2 inhibitor 1)

货号: PC-62409Not For Human Use, Lab Use Only.

MMSET-IN-1 (NSD2 inhibitor 1) is a potent, selective epigenetic oncogene MMSET (aka NSD2 or WHSC1) inhibitor with Ki/IC50 of 1.6/3.3 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

MMSET-IN-1 (NSD2 inhibitor 1) is a potent, selective epigenetic oncogene MMSET (aka NSD2 or WHSC1) inhibitor with Ki/IC50 of 1.6/3.3 uM.
MMSET-IN-1 shows sub-micromolar inhibition of SETD2 and promising selectivity against a panel of 13 other KMTs.

物理化学性质&存储条件

分子量	423.474
分子式	C18H29N7O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S)-2-amino-6-((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)-5-(propylamino)hexanoic acid

参考文献

1. Tisi D, et al. ACS Chem Biol. 2016 Nov 18;11(11):3093-3105.

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MMSET-IN-1 (NSD2 inhibitor 1)

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物理化学性质&存储条件

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MMSET-IN-1 (NSD2 inhibitor 1)

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物理化学性质&存储条件

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