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首页-小分子抑制剂&激动剂-GPCR-Neurokinin Receptor-MLE4901
MLE4901

Chemical Structure : MLE4901

CAS No.: 941690-55-7

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MLE4901 (Pavinetant, MLE-4901, AZD-2624, AZD2624)

货号: PC-61237Not For Human Use, Lab Use Only.

Pavinetant (MLE4901, AZD-2624) is a potent, selective, orally active neurokinin 3 (NK3R) antagonist for the treatment of menopausal hot flushes.

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10 mg ￥2980 In stock
25 mg ￥4980 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Pavinetant (MLE4901, AZD-2624) is a potent, selective, orally active neurokinin 3 (NK3R) receptor antagonist for the treatment of menopausal hot flushes.
Pavinetant (MLE4901, AZD-2624) demonstrates drug-like properties with low metabolic turnover rate in vitro and moderate human plasma protein binding.

物理化学性质&存储条件

分子量 459.56
分子式 C26H25N3O3S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-3-(methylsulfonamido)-2-phenyl-N-(1-phenylpropyl)quinoline-4-carboxamide

参考文献

1. Li Y, et al. Xenobiotica. 2010 Nov;40(11):721-9.

2. Skorupskaite K, et al. Neuroendocrinology. 2017 Apr 5. doi: 10.1159/000473893.

3. Prague JK, et al. Lancet. 2017 May 6;389(10081):1809-1820.

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