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首页-小分子抑制剂&激动剂-GPCR-Glucagon Receptor-MK-3577
MK-3577

Chemical Structure : MK-3577

CAS No.: 1019112-29-8

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MK-3577 (MK 3577, MK3577)

货号: PC-70055Not For Human Use, Lab Use Only.

MK-3577 is a potent, oral active glucagon receptor antagonist blocking the glucagon effect for the treatment of T2DM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    MK-3577 is a potent, oral active glucagon receptor antagonist blocking the glucagon effect for the treatment of T2DM.
    MK-3577 inhibits glucagon-mediated cAMP increases in CHO cells expressing the human glucagon receptor with IC50 of 8.3 nM.

    物理化学性质&存储条件

    分子量 521.03
    分子式 C30H30ClFN2O3
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-(4-((1R,2S)-1-(4-chlorophenyl)-1-(7-fluoro-5-methyl-1H-indol-3-yl)pentan-2-yl)benzamido)propanoic acid

    参考文献

    1. Peng JZ, et al. AAPS J. 2014 Nov;16(6):1259-70.

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