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首页-小分子抑制剂&激动剂-Epigenetics-Histone Acetyltransferase (HAT)-MG149
MG149

Chemical Structure : MG149

CAS No.: 1243583-85-8

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MG149 (MG-149)

货号: PC-20867Not For Human Use, Lab Use Only.

MG149 is a selective histone acetyltransferase Tip60 (KAT5) inhibitor with IC50 of 74 uM, with no activity against PCAF and p300.

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25 mg ￥1980 In stock
100 mg ￥4580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

MG149 is a selective histone acetyltransferase Tip60 (KAT5) inhibitor with IC50 of 74 uM, with no activity against PCAF and p300.
MG149 effectively inhibits acetyltransferase activity of nuclear extracts on the histone H3 and H4 at micromolar concentrations.
MG 149 is competitive with Ac-CoA and noncompetitive with the histone substrate.

物理化学性质&存储条件

分子量 340.46
分子式 C22H28O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-(4-heptylphenethyl)-6-hydroxybenzoic acid

参考文献

1. Massimo Ghizzoni, et al. Eur J Med Chem. 2012 Jan;47(1):337-44.

2. García-González R, et al. Cancers (Basel). 2020 Oct 15;12(10):2986.

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