MG-101 |CAS:110044-82-1 Probechem Biochemicals

Chemical Structure : MG-101

CAS No.: 110044-82-1

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MG-101 (Calpain inhibitor I, ALLN, MG101)

货号: PC-45577Not For Human Use, Lab Use Only.

MG-101 (ALLN) is a potent inhibitor of cysteine proteases including calpain I (Ki= 190 nM), calpain II (Ki= 220 nM), cathepsin B (Ki= 150 nM) and cathepsin L (Ki= 500 pM).

规格	价格	库存
10 mg	￥880	In stock
25 mg	￥1580	In stock
50 mg	￥2580	In stock
100 mg		Get quote

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生物&药学活性

MG-101 (ALLN) is a potent inhibitor of cysteine proteases including calpain I (Ki= 190 nM), calpain II (Ki= 220 nM), cathepsin B (Ki= 150 nM) and cathepsin L (Ki= 500 pM).
MG-101 activates p53-dependent apoptosis in tumor cell lines.
MG-101 increases activated p53, p21 and caspase levels and promotes cell cycle arrest through inhibition of cyclin D degradation in vitro.

物理化学性质&存储条件

分子量	383.5255
分子式	C20H37N3O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	L-Leucinamide, N-acetyl-L-leucyl-N-[(1S)-1-formylpentyl]-

参考文献

1. Zhang L, et al. J Biol Chem. 1999 Mar 26;274(13):8966-72.

2. Inoue S,et al. J Biol Chem. 1991 Jul 15;266(20):13311-7.

3. Sherwood SW, et al. Proc Natl Acad Sci U S A. 1993 Apr 15;90(8):3353-7.

MG-101 (Calpain inhibitor I, ALLN, MG101)

生物&药学活性

物理化学性质&存储条件

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MG-101 (Calpain inhibitor I, ALLN, MG101)

生物&药学活性

物理化学性质&存储条件

参考文献

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