MDL100907 (Volinanserin) | 5-HT2A antagonist | Probechem Biochemicals

Chemical Structure : MDL100907

CAS No.: 139290-65-6

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MDL100907 (MDL-100907, Volinanserin)

货号: PC-60814Not For Human Use, Lab Use Only.

MDL100907 (Volinanserin) is a potent, selective 5-HT2A receptor antagonist with Ki of 0.36 nM, > 80-fold selectivity for 5-HT2A over other serotonergic receptors.

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10 mg	￥1480	In stock
25 mg	￥2580	In stock
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生物&药学活性

MDL100907 (Volinanserin) is a potent, selective 5-HT2A receptor antagonist with Ki of 0.36 nM, > 80-fold selectivity for 5-HT2A over other serotonergic receptors.
MDL100907 demonstrates a clozapine-like profile of potential antipsychotic activity with low extrapyramidal sid-effect liability, and has a superior CNS safety index.

物理化学性质&存储条件

分子量	373.46
分子式	C22H28FNO3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-(+)-α-(2,3-Dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperinemethanol

参考文献

1. Ardayfio PA, et al. J Pharmacol Exp Ther. 2008 Dec;327(3):891-7.

2. Sorensen SM, et al. J Pharmacol Exp Ther. 1993 Aug;266(2):684-91.

3. Kehne JH, et al. J Pharmacol Exp Ther. 1996 May;277(2):968-81.

MDL100907 (MDL-100907, Volinanserin)

生物&药学活性

物理化学性质&存储条件

参考文献

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MDL100907 (MDL-100907, Volinanserin)

生物&药学活性

物理化学性质&存储条件

参考文献

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