MCT1-IN-4a |CAS:1448314-00-8 Probechem Biochemicals

Chemical Structure : MCT1-IN-4a

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MCT1-IN-4a

货号: PC-62725Not For Human Use, Lab Use Only.

MCT1-IN-4a is a potent, selective monocarboxylate transporter 1 (MCT1) inhibitor with IC50 of 90 nM.

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生物&药学活性

MCT1-IN-4a is a potent, selective monocarboxylate transporter 1 (MCT1) inhibitor with IC50 of 90 nM; exhibits significant single agent activity in MCT1 expressing GL261-luc2 syngraft model, but not in MCT4 expressing MDA-MB-231 xenograft model; has good absorption, metabolic stability, and a low drug efflux ratio.

物理化学性质&存储条件

分子量	385.419
分子式	C24H19NO4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	7-(dibenzylamino)-2-oxo-2H-chromene-3-carboxylic acid

参考文献

1. Gurrapu S, et al. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3282-6.

MCT1-IN-4a

生物&药学活性

物理化学性质&存储条件

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MCT1-IN-4a

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