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首页-小分子抑制剂&激动剂-GPCR-Melanocortin Receptor-MCL0020
MCL0020

Chemical Structure : MCL0020

CAS No.: 475498-26-1

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MCL0020 (MCL 0020)

货号: PC-21480Not For Human Use, Lab Use Only.

MCL0020 is a potent, selective inverse agonist of melanocortin MC4 receptor (MC4R) with binding IC50 of 11.6 nM, shows negligible affinity for MC1 and MC3 receptors.

规格 价格 库存 数量
2 mg ￥2480 In stock
5 mg ￥3980 In stock
10 mg ￥5880 In stock
25 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

MCL0020 is a potent, selective inverse agonist of melanocortin MC4 receptor (MC4R) with binding IC50 of 11.6 nM, shows negligible affinity for MC1 and MC3 receptors.
MCL0020 attenuates swim stress-induced anxiogeniclike behavior in light/dark exploration tests in mice, significantly reverses stress-induced anorexia in rats.

物理化学性质&存储条件

分子量 609.72
分子式 C34H39N7O4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N-Acetyl-3-(2-naphthalenyl)-D-alanyl-L-arginyl-3-(2-naphthalenyl)-L-alaninamide

参考文献

1. Chaki S, et al. Eur J Pharmacol. 2003 Aug 1;474(1):95-101.

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