Linagliptin |CAS:668270-12-0 Probechem Biochemicals

Chemical Structure : Linagliptin

CAS No.: 668270-12-0

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Linagliptin (BI 1356;BI-1356;BI1356)

货号: PC-42508Not For Human Use, Lab Use Only.

Linagliptin (BI-1356) is a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM.

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25 mg	￥880	In stock
100 mg	￥1580	In stock
200 mg	￥2480	In stock
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生物&药学活性

Linagliptin (BI-1356) is a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM.
Linagliptin (BI-1356) shows no significant inhibition on hERG and muscarinic receptor M1 at 1 uM.
Linagliptin (BI-1356) shows considerable blood glucose lowering in different animal species.

物理化学性质&存储条件

分子量	472.5422
分子式	C25H28N8O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1H-Purine-2,6-dione, 8-[(3R)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-

参考文献

1. Eckhardt M, et al. J Med Chem. 2007 Dec 27;50(26):6450-3.

2. Thomas L, et al. J Pharmacol Exp Ther. 2008 Apr;325(1):175-82.

3. Thomas L, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):556-63.

Linagliptin (BI 1356;BI-1356;BI1356)

生物&药学活性

物理化学性质&存储条件

参考文献

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Linagliptin (BI 1356;BI-1356;BI1356)

生物&药学活性

物理化学性质&存储条件

参考文献

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