Legumain inhibitor 10t

Chemical Structure : Legumain inhibitor 10t

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货号: PC-20813Not For Human Use, Lab Use Only.

Legumain inhibitor 10t is a potent, selective and cellularly active Legumain (asparagine endopeptidase, AEP) inhibitor with IC50 of 71 nM.

规格	价格	库存	数量
50 mg		Get quote
100 mg		Get quote
200 mg		Get quote
1 g		Get quote

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生物&药学活性

Legumain inhibitor 10t is a potent, selective and cellularly active Legumain (asparagine endopeptidase, AEP) inhibitor with IC50 of 71 nM.
Legumain inhibitor 10t blocks colony formation in both metastatic breast (MCF7) and prostate (PC3) cancer cell lines with IC50 of 5 and 2.5 uM, respectively.

物理化学性质&存储条件

分子量	482.60
分子式	C25H30N4O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C([C@H]1N(S(=O)(C2=CC=C(C3=CC=C(C(C)(C)C)C=C3)C=C2)=O)CCC1)N[C@H](C#N)CC(N)=O

参考文献

1. Kerry A Ness, et al. Bioorg Med Chem Lett. 2015 Dec 1;25(23):5642-5.