LY3027788 | mGlu2/3 antagonist | Probechem Biochemicals

Chemical Structure : LY3027788

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LY3027788 (LY-3027788, LY 3027788)

货号: PC-60731Not For Human Use, Lab Use Only.

LY3027788 is an orally active prodrug of LY3020371, which is a potent, selective metabotropic glutamate 2/3 receptor (mGlu2/3) antagonist with Ki of 5.3 and 2.5 nM, respectively.

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生物&药学活性

LY3027788 is an orally active prodrug of LY3020371, which is a potent, selective metabotropic glutamate 2/3 receptor (mGlu2/3) antagonist with Ki of 5.3 and 2.5 nM, respectively.
LY3027788 augments the antidepressant-like effects of fluoxetine or citalopram without altering plasma or brain levels of these compounds.

物理化学性质&存储条件

分子量	591.576
分子式	C25H31F2NO11S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	bis(((isopropoxycarbonyl)oxy)-methyl) (1S,2R,3S,4S,5R,6R)-2-amino-3-(((3,4-difluorophenyl)thio)methyl)-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylate

参考文献

1. Witkin JM, et al. J Pharmacol Exp Ther. 2017 Apr;361(1):68-86.

LY3027788 (LY-3027788, LY 3027788)

生物&药学活性

物理化学性质&存储条件

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LY3027788 (LY-3027788, LY 3027788)

生物&药学活性

物理化学性质&存储条件

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