LY2318912 |CAS:874902-18-8 Probechem Biochemicals

Chemical Structure : LY2318912

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LY2318912 (LY 2318912)

货号: PC-63017Not For Human Use, Lab Use Only.

LY2318912 is a potent, competitive, small molecule inhibitor of anandamide uptake with IC50 of 7.27 nM, shows high affinity against anandamide transporter binding site with Kd of 7.62 nM.

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生物&药学活性

LY2318912 is a potent, competitive, small molecule inhibitor of anandamide uptake with IC50 of 7.27 nM, shows high affinity against anandamide transporter binding site with Kd of 7.62 nM.
LY2318912 elevates anandamide levels 5-fold in the brain and demonstrates efficacy in the formalin paw-licking model of persistent pain with no obvious adverse effects on motor function in rodents.

物理化学性质&存储条件

分子量	441.193
分子式	C12H12IN9O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-[(4-azido-3-iodo-benzoylamino)-methyl]-tetrazole-1-carboxylic acid dimethylamide

参考文献

1. Moore SA, et al. Proc Natl Acad Sci U S A. 2005 Dec 6;102(49):17852-7.

2. Ortar G, et al. Eur J Med Chem. 2008 Jan;43(1):62-72.

LY2318912 (LY 2318912)

生物&药学活性

物理化学性质&存储条件

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LY2318912 (LY 2318912)

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