LUF6000 |CAS:890087-21-5 Probechem Biochemicals

Chemical Structure : LUF6000

CAS No.: 890087-21-5

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LUF6000 (LUF-6000;LUF 6000)

货号: PC-43415Not For Human Use, Lab Use Only.

LUF6000 is a potent, selective, positive allosteric modulator (enhancer) of human A3 adenosine receptor, enhance Emax but without affecting agonist potency.

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5 mg	￥2480	In stock
10 mg	￥3980	In stock
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LUF6000 is a potent, selective, positive allosteric modulator (enhancer) of human A3 adenosine receptor, enhance Emax but without affecting agonist potency.
LUF6000 enhance sagonist efficacy in a functional assay by 45% and decreases dissociation rate similarly without influencing agonist potency.
LUF6000 is superior to that of DU124183.

物理化学性质&存储条件

分子量	411.327
分子式	C22H20Cl2N4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3H-Imidazo[4,5-c]quinolin-4-amine, 2-cyclohexyl-N-(3,4-dichlorophenyl)-

参考文献

1. Göblyös A, et al. J Med Chem. 2006 Jun 1;49(11):3354-61.

2. Gao ZG, et al. BMC Pharmacol. 2008 Dec 12;8:20.

3. Gao ZG, et al. Biochem Pharmacol. 2011 Sep 15;82(6):658-68.

LUF6000 (LUF-6000;LUF 6000)

生物&药学活性

物理化学性质&存储条件

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LUF6000 (LUF-6000;LUF 6000)

生物&药学活性

物理化学性质&存储条件

参考文献

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