LUF5834 | A2AR agonist | Probechem Biochemicals

Chemical Structure : LUF5834

加入收藏

LUF5834 (LUF-5834)

货号: PC-22361Not For Human Use, Lab Use Only.

LUF5834 is a potent, selective, non-adenosine adenosine A1 receptor adenosine receptor (A2BR) partial agonist with EC50 of 12 nM (hA2B), 45-fold selective over hA3, also shows high affinity with Ki of 2.6 nM and 28 nM for hA1 and hA2A, respectively.

规格	价格	库存	数量
5 mg		Get quote
10 mg		Get quote
25 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

LUF5834 is a potent, selective, non-adenosine adenosine A1 receptor adenosine receptor (A2BR) partial agonist with EC50 of 12 nM (hA2B), 45-fold selective over hA3.
LUF5834 also shows high affinity with Ki of 2.6 nM and 28 nM for hA1 and hA2A, respectively.

物理化学性质&存储条件

分子量	348.38
分子式	C17H12N6OS
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-amino-4-(4-hydroxyphenyl)-6-(1H-imidazol-2-ylmethylsulfanyl)pyridine-3,5-dicarbonitrile

参考文献

1. Beukers MW, et al. J Med Chem. 2004 Jul 15;47(15):3707-9.

2. Urmaliya VB, et al. J Cardiovasc Pharmacol. 2009 May;53(5):424-33.

3. Lane JR, et al. Biochem Pharmacol. 2010 Oct 15;80(8):1180-9.

LUF5834 (LUF-5834)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

LUF5834 (LUF-5834)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.