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首页-小分子抑制剂&激动剂-Epigenetics-Histone Methyltransferase (HMTase)-LH168
LH168

Chemical Structure : LH168

CAS No.:

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LH168 (LH-168)

货号: PC-25506Not For Human Use, Lab Use Only.

LH168 is a potent, exquisitely selective WDR5 chemical probe inhibitor with EC50 of 10 nM in cellulo target engagement NanoBRET assays, SPR KD of 1.9 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

LH168 is a potent, exquisitely selective WDR5 chemical probe inhibitor with EC50 of 10 nM in cellulo target engagement NanoBRET assays, SPR KD of 1.9 nM.

物理化学性质&存储条件

分子量 584.66
分子式 C29H31F3N6O2S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-3-((1H-imidazol-1-yl)methyl)-N-(1-(6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-1-oxopentan-2-yl)-5-(1-ethyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)benzamide

参考文献

1. Lasse Hoffmann, et al. RSC Chem Biol. 2025 Jul 17. doi: 10.1039/d5cb00109a.

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