LGD-3303 |CAS:917891-35-1 Probechem Biochemicals

Chemical Structure : LGD-3303

CAS No.: 917891-35-1

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LGD-3303 (LGD3303)

货号: PC-61861Not For Human Use, Lab Use Only.

LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.

规格	价格	库存
10 mg	￥1280	In stock
25 mg	￥1980	In stock
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100 mg		Get quote

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生物&药学活性

LGD-3303 is an orally available, brain-penetrant nonsteroidal selective androgen receptor modulator (SARM) that that shows little or no cross-reactivity with related nuclear receptors.
LGD-3303 has potent activity on levator ani muscle but is a partial agonist on the preputial gland and ventral prostate in a castrated rat model of androgen deficiency。
LGD-3303 enhances male-directed sexual preference, proceptive behavior, and lordosis behavior in sexually experienced, but not sexually naive, female rats.

物理化学性质&存储条件

分子量	342.743
分子式	C16H14ClF3N2O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	9-Chloro-2-ethyl-1-methyl-3-(2,2,2-trifluoroethyl)-3H-pyrrolo(3,2-F)quinolin-7(6H)-one

参考文献

1. Vajda EG, et al. J Pharmacol Exp Ther. 2009 Feb;328(2):663-70.

2. Vajda EG, et al. J Bone Miner Res. 2009 Feb;24(2):231-40.

3. Kudwa AE, et al. Endocrinology. 2010 Jun;151(6):2659-68.

LGD-3303 (LGD3303)

生物&药学活性

物理化学性质&存储条件

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LGD-3303 (LGD3303)

生物&药学活性

物理化学性质&存储条件

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