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首页-小分子抑制剂&激动剂-GPCR-Cannabinoid Receptor-LEI-102
LEI-102

Chemical Structure : LEI-102

CAS No.: 1228659-40-2

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LEI-102 (LEI 102)

货号: PC-20746Not For Human Use, Lab Use Only.

LEI-102 (LEI 102) is a potent, selective cannabinoid CB2 receptor agonist with binding pKi of 8.0, 1000-fold selectivity over CB1R.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

LEI-102 (LEI 102) is a potent, selective cannabinoid CB2 receptor agonist with binding pKi of 8.0, 1000-fold selectivity over CB1R.
LEI-102 is more potent than the selective CB2R agonists APD371 and HU308.
LEI-102 activates CB2R as a partial agonist (Emax 76 ± 1%) with a pEC50 value of 6.9 in G protein activation assays.

物理化学性质&存储条件

分子量 454.55
分子式 C25H31FN4O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

O=C1N(CC(C)C)C(CN1CC2=CC=C(C3=NC(CNC4CCOCC4)=C(F)C=C3)C=C2)=O

参考文献

1. Xiaoting Li, et al. Nat Commun. 2023 Mar 15;14(1):1447.

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