KT5720

Chemical Structure : KT5720

CAS No.: 108068-98-0

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货号: PC-23453Not For Human Use, Lab Use Only.

KT5720 is a potent, cell-permeable, specific, reversible and ATP-competitive PKA inhibitor with IC50 of 3.3 uM.

规格	价格	库存
50 ug	￥1380	In stock
100 ug	￥2380	In stock
500 ug	￥5980	In stock
1 mg		Get quote

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生物&药学活性

KT5720 is a potent, cell-permeable, specific, reversible and ATP-competitive PKA inhibitor with IC50 of 3.3 uM.
KT5720 is effective in reversing MDR1-mediated multidrug resistance.
KT5720 also reduces the excitability of dorsal root ganglion (DRG) neurons by attenuating Hyperpolarization-activated cyclic nucleotide-gated (HCN) channel activity and reducing intracellular Ca2+ concentrations.

物理化学性质&存储条件

分子量	537.62
分子式	C32H31N3O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	9,12-Epoxy-1H-diindolo[1,2,3-fg:3′,2′,1′-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid, 2,3,9,10,11,12-hexahydro-10-hydroxy-9-methyl-1-oxo-, hexyl ester, (9R,10S,12S)-

参考文献

1. Davies SP, et al. Biochem J. 2000 Oct 1;351(Pt 1):95-105.

2. Galski H, et al. Leuk Res. 2006 Sep;30(9):1151-8.

KT5720

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物理化学性质&存储条件

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KT5720

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