KI-MS2-008

Chemical Structure : KI-MS2-008

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货号: PC-20800Not For Human Use, Lab Use Only.

KI-MS2-008 is a small molecule Max binder that modulate Myc-driven transcription in cells (IC50=1.28 uM) and inhibit viable cell levels in a Myc-dependent manner.

规格	价格	库存	数量
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200 mg		Get quote

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生物&药学活性

KI-MS2-008 is a small molecule Max binder that modulate Myc-driven transcription in cells (IC50=1.28 uM) and inhibit viable cell levels in a Myc-dependent manner.
KI-MS2-008 induces Max/Max homodimerization.
KI-MS2-008 (10 uM) decreases Myc protein levels and affects the global Myc transcriptional program in ST486 cells.
KI-MS2-008 also decreases viable cancer cell growth in a Myc-dependent manner and suppresses tumor growth in vivo.

物理化学性质&存储条件

分子量	536.65
分子式	C32H28N2O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(3aS,10bS)-3a-benzyl-2-phenyl-5-(2-(phenylsulfonyl)ethyl)-3a,5,6,10b-tetrahydro-4H-benzo[c]oxazolo[5,4-e]azepin-4-one

参考文献

1. Struntz NB, et al. Cell Chem Biol. 2019 May 16;26(5):711-723.e14.

KI-MS2-008

生物&药学活性

物理化学性质&存储条件

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KI-MS2-008

生物&药学活性

物理化学性质&存储条件

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