KDM5A covalent inhibitor N73 |CAS 2288785-06-6 Probechem Biochemicals

Chemical Structure : KDM5A covalent inhibitor N73

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KDM5A covalent inhibitor N73 (KDM5A inhibitor N73)

货号: PC-35801Not For Human Use, Lab Use Only.

KDM5A covalent inhibitor N73 is the the isopropyl ester derivative of N71, an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481, >20-fold selectivity over KDM4A..

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KDM5A covalent inhibitor N73 is the the isopropyl ester derivative of N71, an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481, >20-fold selectivity over KDM4A.

物理化学性质&存储条件

分子量	564.745
分子式	C31H40N4O4S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	isopropyl (E)-2-((3-(4-(dimethylamino)but-2-enamido)phenyl)(2-(piperidin-1-yl)ethoxy)methyl)thieno[3,2-b]pyridine-7-carboxylate

参考文献

1. Horton JR, et al. J Med Chem. 2018 Nov 15. doi: 10.1021/acs.jmedchem.8b01219.

KDM5A covalent inhibitor N73 (KDM5A inhibitor N73)

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KDM5A covalent inhibitor N73 (KDM5A inhibitor N73)

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